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Department of Organic Chemistry

Faculty of Pharmacy

PUBLICATION ACTIVITIES

Main publications:

  1. Fedorowicz, J, Sączewski, J., Drażba, Z., Wiśniewska, P., Gdaniec, M., Wicher, B., Suwiński, G., Jalińska, A.
    Synthesis and fluorescence of dihydro-[1,2,4]triazolo[4,3-a]pyridin-2-ium-carboxylates: An experimental and TD-DFT comparative study;
    Dyes and Pigments 161 (2019), p. 347-359,
    (go to article)
  2. Fedorowicz, J., Sączewski, J., Konopacka, A., Waleron, K., Lejnowski, D., Ciura, K., Tomašič, T., Skok, Ž., Savijoki, K., Morawska, M.,Gilbert-Girard, S., Fallarero, A.
    Synthesis and biological evaluation of hybrid quinolone-based quaternary ammonium antibacterial agents;
    European Journal of Medicinal Chemistry 179, (2019), pp. 576-590,
    (go to article)
  3. Fedorowicz, J., Gzella, K., Wiśniewska, P., Sączewski, J.
    2,2’-[(1,4-dimethoxy-1,4-dioxobutane-2,3-diylidene)bis(azanylylidene)]bis(quinoline-3-carboxylic acid);
    MolBank. (2019), Article number M1093
    (go to article)
  4. Makowska, A., Saczewski, F., Bednarski, P.J., Saczewski, J., Balewski, Ł.
    Hybrid molecules composed of 2,4-diamino-1,3,5-triazines and 2-imino-coumarins and coumarins. Synthesis and cytotoxic properties;
    Molecules. 23 (2018), 1616,
    (go to article)
  5. Mazur, L., Saczewski, J., Jarzembska, K.N., Szwarc-Karabyka, K., Paprocka, R., Modzelewska-Banachiewicz, B.;
    Synthesis, structural characterization and reactivity of new trisubstituted: N 1-acylamidrazones: Solid state and solution studies;
    CrystEngComm. 20 (2018), 4179-4193,
    (go to article)
  6. Fedorowicz, J., Sączewski, J.
    Modifications of quinolones and fluoroquinolones: hybrid compounds and dual-action molecules;
    Monatshefte fur Chemie. 149 (2018), 1199-1245,
    (go to article)
  7. Krause, M., Foks, H., Augustynowicz-Kopeć, E., Napiórkowska, A., Szczesio, M., Gobis, K.
    Synthesis and tuberculostatic activity evaluation of novel benzazoles with alkyl, cycloalkyl or pyridine moiety;
    Molecules. 23 (2018), 985,
    (go to article)
  8. Szczesio, M., Gołka, J., Korona-Głowniak, I.,Gobis, K.,
    Planarity of benzoyldithiocarbazate tuberculostatics.V antibacterial activities of diesters of benzoyldithiocarbazic acid;
    Journal of Molecular Structure. 1167 (2018), 127-133,
    (go to article)
  9. Szczesio, M., Gołka, J., Korona-Głowniak, I., Orlewska, C., Gobis, K., Olczak, A.
    Planarity of heteroaryldithiocarbazic acid derivatives showing tuberculostatic activity: Structure-activity relationships;
    Acta Crystallographica Section C: Structural Chemistry. 74 (2018), 400-405,
    (go to article)
  10. Główka M.L., Kałużyńska S., Krause, M., Gobis, K., Foks, H., Szczesio, M., Olczak, A ;
    SThe structures of benzimidazole derivatives and their potential as tuberculostatics;
    Acta Crystallographica Section C: Structural Chemistry. 74 (2018), 1684-1691,
    (go to article)
  11. Pogorzelska A., Żołnowska B., Bartoszewski R.;
    Cysteine cathepsins as a prospective target for anticancer therapies—current progress and prospects;
    Biochimie 151 (2018) 85-106,
    (go to article)
  12. Kawczak P., Belka M, Sławiński J, Bączek T.;
    QSRR evaluation of the new anticancer sulfonamides in view of the cis-trans isomerism
    Current Pharmaceutical Analysis 14 (2018) 35-40,
    (go to article)
  13. Pogorzelska A., Żołnowska B., Sławiński J., Kawiak A., Szafrański K., Belka M., Bączek T.;
    Synthesis of 2-alkylthio-N-(quinazolin-2-yl)benzenesulfonamide derivatives: anticancer activity, QSAR studies, and metabolic stability;
    Monatshefte fur Chemie 149 (2018) 1885-1898,
    (go to article)
  14. Pogorzelska A., Sławiński J., Kawiak A., Żołnowska B., Chojnacki J.,, Stasiłojć G., Ulenberg S., Szafrański K., Bączek T.; ISynthesis, molecular structure, and metabolic stability of new series of N’-(2-alkylthio-4-chloro-5-methylbenzenesulfonyl)-1-(5-phenyl-1H-pyrazol-1-yl)amidine as potential anti-cancer agents; European Journal of Medicinal Chemistry 155 (2018) 670-680, (go to article)
  15. Zuvela P., Liu J., Myunggi Y., Pomastowski P., Sagandykova G., Belka M., David J., Bączek T., Krzysztof Szafrański, Beata Żołnowska, Jarosław Sławiński, Supuran C., Wong M., Buszewski B.; Target-based drug discovery through inversion of quantitative structure-drug property relationships and molecular simulation: CA IX-sulphonamide complexes. J. Enz. Inhib. Med. Chem. 33 (2018) 1430‒1443; (go to article)
  16. Cieślik P., Woźniak M., Tokarski K., Kusek M., Pilca A., Płoska A., Radulska A., Pelikant-Małecka I, Beata Żołnowska, Jarosław Sławiński, Kalinowski L., Wierońska J.; Simultaneous activation of muscarinic and GABAB receptors as a bidirectional target for novel antipsychotic. Behav. Brain Res. (2018), (go to article)
  17. Żołnowska, B.; Sławiński, J.; Brzozowski, Z.; Kawiak, A.; Belka, M.; Zielińska, J.; Baczek˛, T.; Chojnacki, J. Synthesis, molecular structure, anticancer activity, and QSAR study of N-(Aryl/heteroaryl)-4-(1h-pyrrol-1-yl)benzenesulfonamide derivatives. Int. J. Mol. Sci. 2018, 19, 1–23, (go to article)
  18. Monti, S. M.; Meccariello, A.; Ceruso, M.; Szafrański, K.; Sławiński, J.; Supuran, C. T. Inhibition studies of Brucella suis β-carbonic anhydrases with a series of 4-substituted pyridine-3-sulphonamides. J. Enzyme Inhib. Med. Chem. 2018, 33, (go to article)
  19. Żołnowska B., Sławiński J, Szafrański K., Angeli A, Supuran C.T., Kawiak A., Wieczór M., Zielińska J., Bączek T.; Novel 2-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)-1-(1,3,5-triazin-2-ylamino)guanidine derivatives: Inhibition of human carbonic anhydrase cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII, anticancer activity, and molecular modeling studies; European Journal of Medicinal Chemistry 143 (2018) 1931-1941, (go to article)
  20. Szafrański K., Sławiński J., Kędzia A., Kwapisz E.; Syntheses of Novel 4-Substituted N-(5-amino-1H-1,2,4-triazol-3-yl)pyridine-3-sulfonamide Derivatives with Potential Antifungal Activity; Molecules 22 (11) (2017), art 1926, (go to article)
  21. Pogorzelska A., Żołnowska B., Sławiński J., Szafrański K., Kawiak A., Chojnacki J., Ulenberg S., Zielińska J.,Bączek T.; Novel 2-(2-alkylthiobenzenesulfonyl)-3-(phenylprop-2-ynylideneamino)guanidine derivatives as potent anticancer agents – Synthesis, molecular structure, QSAR studies and metabolic stability; European Journal of Medicinal Chemistry 138 (2017) 357-370, (go to article)
  22. J. Sączewski, J. Fedorowicz, M. Gdaniec, P. Wiśniewska, E. Sieniawska, Z.Drażba, J. Rzewnicka, Ł. Balewski ; The Elusive Paal–Knorr Intermediates in the Trofimov Synthesis of Pyrroles: Experimental and Theoretical Studies; Journal of Organic Chemistry. 82, 2017, 9737-9743(go to article)
  23. Sławiński J., Szafrański K., Pogorzelska A., Żołnowska B., Kawiak A., Macur K., Belka M., Bączek T.; Novel 2-benzylthio-5-(1,3,4-oxadiazol-2-yl)benzenesulfonamides with anticancer activity: Synthesis, QSAR study, and metabolic stability; European Journal of Medicinal Chemistry 132 (2017) 236-248, (go to article)
  24. Zołnowska B., Sławiński J., Pogorzelska A., Szafrański K., Kawiak A., Stasiłojć G., Belka M., Zielińska J., Bączek T.; Synthesis, QSAR studies, and metabolic stability of novel 2-alkylthio-4-chloro-N-(5-oxo-4,5-dihydro-1,2,4-triazin-3-yl)benzenesulfonamide derivatives as potential anticancer and apoptosis-inducing agents; Chem Biol Drug Des. 2017;1–17. (go to article)
  25. Zołnowska B., Sławiński J., Pogorzelska A., Szafrański K., Kawiak A., Stasiłojć G., Belka M., Ulenberg S., Baczek T., Chojnacki J. Novel 5-substituted 2-(aylmethylthio)-4-chloro-N-(5-aryl-1,2,4-triazin-3-yl)benzenesulfonamides: Synthesis, molecular structure, anticancer activity, apoptosis-inducing activity and metabolic stability(Article) Molecules 21 (1) (2016), art 808, (go to article)
  26. J. Sławiński, A. Grzonek, B. Żołnowska, A. Kawiak; Synthesis of novel pyrido[4,3-e][1,2,4]triazino[3,2-c][1,2,4]thiadiazine 6,6-dioxide derivatives with potential anticancer activity; Molecules 21 (1) (2016), art 41, s. 1-16 (go to article)
  27. A. Pogorzelska, J. Sławiński, K. Brożewicz, Sz. Ulenberg, T. Bączek; Novel 3-Amino-6-chloro-7-(azol-2 or 5-yl)-1,1-dioxo-1,4,2-benzodithiazine Derivatives with Anticancer Activity: Synthesis and QSAR Study; Molecules 20(12) (2015), 21960-21970 (go to article)
  28. B. Żołnowska, J. Sławiński, A. Grzonek, A. Kędzia, E. Kwapisz, A. Kawiak; N-Substituted N′-(2-alkylthio-4-chloro-5-methylbenzenesulfonyl)guanidines – Antibacterial, Cytotoxic Activities and Some Structure-Activity Relationships; Pol. J. Microbiol. 63 (3) 2015 299-305; (go to article)
  29. B. Żołnowska, J. Sławiński, M. Belka, T. Bączek, A. Kawiak, J. chojnacki, A. Pogorzelska, K. Szafrański Synthesis, Molecular Structure, Metabolic Stability and QSAR Studies of a Novel Series of Anticancer N-Acylbenzenesulfonamides; Molecules 20(10) 2015, 19101-19129; (go to article)
  30. J. Sączewski, J. Fedorowicz, M. Korcz, F. Sączewski, B. Wicher, M. Gdaniec, A. Konopacka; Experimental and theoretical studies on the tautomerism and reactivity of isoxazolo[3,4-b]quinolin-3(1H)-ones; Tetrahedron. 2015; (go to article)
  31. A. Bułakowska, M. Konieczny; Synthesis of vinyl sulfones by ring opening of 4,4-dioxo-2,3-dihydrobenzo[b][1,4]oxathiines and their in situ reactions with nucleophilic or electrophilic agents; J. Het. Chem. 2015; vol. 52, nr 2, s. 440-444; (go to article)
  32. M. Konieczny, A. Bułakowska, D. Pirska, W. Konieczny, A. Składanowski, M. Sabisz, M. Wojciechowski, K. Lemke, A. Pieczykolan, W. Strożek, Structural factors affecting affinity of cytotoxic oxathiole-fused chalcones toward tubulin, Eur. J. Med. Chem. 2015; vol. 89, s. 733-742 (go to article)
  33. I. Łącka, M. Konieczny, A. Bułakowska, M. Kodedová, D. Gašková, I. K. Maurya, R. Prasad, S. Milewski, Chemosensitization of multidrug resistant Candida albicans by the oxathiolone fused chalcone derivatives, Front. Microbiol. 2015; vol. 6, art. 783 (go to article)
  34. K. Gobis H. Foks,M. Serocki, E. Augustynowicz-Kopeć, A. Napiórkowska ;Synthesis and evaluation of in vitro antimycobacterial activity of novel 1H-benzo[d]imidazole derivatives and analogues ; Eur. J. Med. Chem. 89 (2015), 13-20,
    (go to article)
  35. K.Szafrański, J. Sławiński, Synthesis of Novel 1-(4-Substituted pyridine-3-sulfonyl)-3-phenylureas with Potential Anticancer Activity; Molecules 20(7) 2015, 12029-12044 (go to full text)
  36. K. Gobis H. Foks, K. Suchan, E. Augustynowicz-Kopeć, A. Napiórkowska, K. Bojanowski ; Novel 2-(2-phenalkyl)-1H-benzo[d]imidazoles as antitubercular agents. Synthesis, biological evaluation and structure-activity relationship; Bioorg. Med. Chem. 23 (2015), 2112–2120,
    (go to article)
  37. J. Sławiński, B. Żołnowska, Z. Brzozowski, A. Kawiak, M. Belka, T. Bączek Synthesis and QSAR Study of Novel 6-Chloro-3-(2-Arylmethylene-1-methylhydrazino)-1,4,2-benzodithiazine 1,1-Dioxide Derivatives with Anticancer Activity; Molecules 20(4) 2015, 5754-5770 (go to full text)
  38. M.. Konieczny, A. Bułakowska, J. Polak, D. Pirska, W. Konieczny, P. Gryń, A. Składanowski, M. Sabisz, K. Lemke, A. Pieczykolan, M. Gałązka, K. Wiciejowska, J. Wietrzyk, Structural factors affecting cytotoxic activity of (E)-1-(benzo[d ][1,3]oxathiol-6-yl)-3-phenylprop-2-en-1-one derivatives, Chem. Biol. Drug Des. 2014; vol. 84, nr 1, 86-91 (go to article)
  39. B. Żołnowska, J. Sławiński, A. Pogorzelska, J. Chojnacki, D. Vullo, C.T. Supuran; Carbonic anhydrase inhibitors. Synthesis, and molecular structure of novel series N-substituted N′-(2-arylmethylthio-4-chloro-5- methylbenzenesulfonyl)guanidines and their inhibition of human cytosolic isozymes i and II and the transmembrane tumor-associated isozymes IX and XII; Eur. J. Med. Chem. 71 (2014), 135-147. (go to article)
  40. J. Sławiński, A. Pogorzelska, B. Żołnowska, A. Kędzia, M. Ziółkowska-Klinkosz, E. Kwapisz; Synthesis and Anti-Yeast Evaluation of Novel 2-Alkylthio-4-chloro-5-methyl-N-[imino-(1-oxo-(1H)-phthalazin-2-yl)methyl]benzenesulfonamide Derivatives; Molecules 19 (2014), 13704-13723 (go to article)
  41. E. Sikorska, M. Dawgul, K. Greber, E. Iłowska, A. Pogorzelska, W. Kamysz; Self-assembly and interactions of short antimicrobial cationic lipopeptides with membrane lipids: ITC, FTIR and molecular dynamics studies;BBA-Biomembranes 2625-2635. (go to article)
  42. M. Belka, W. Hewelt-Belka, J. Sławiński, T.Bączek; Mass Spectrometry Based Identification of Geometric Isomers during Metabolic Stability Study of a New Cytotoxic Sulfonamide Derivatives Supported by Quantitative Structure-Retention Relationships; PLOS ONE 9 (2014), e98096. (go to article)
  43. M. Konieczny, A. Bułakowska, J. Polak, D. Pirska, W. Konieczny, P. Gryń, A. Skladanowski, M. Sabisz, K. Lemke, A. Pieczykolan, M. Gałązka, K. Wiciejowska, J. Wietrzyk; Structural Factors Affecting Cytotoxic Activity of (E)-1-(Benzo[d ][1,3]oxathiol-6-yl)-3-phenylprop-2-en-1-one Derivatives; Chem. Biol. Drug Des. 84 (2014), 86-91. (go to article)
  44. J. Sączewski, A. Kędzia, A. Jalińska; New derivatives of 4,6-dimethylisoxazolo[3,4-b] pyridin-3(1H)-one: synthesis, tautomerism, electronic structure and antibacterial activity; Heterocycl. Commun. 51 (2014), 215-223. (go to article)
  45. J. Sączewski, M. Korcz; Synthesis and reactivity of heterocyclic hydroxylamine-O-sulfonates; Heterocycl. Commun. 51 (2014), 133-147.
    (go to article)
  46. H. Foks, D. Pancechowska-Ksepko, K. Gobis; Synthesis and Characterization of Novel N-Alkylamine- and N-Cycloalkylamine-Derived 2-Benzoyl-N-aminohydrazinecarbothioamides, 1,3,4-Thiadiazoles and 1,2,4-Triazole-5(4H)thiones; J. Het. Chem. 51 (2014), 98-105,
    (go to article)
  47. R. Hałasa, K. Turecka, Cz. Orlewska, W. Werel; Comparison of fluorescence optical respirometry and microbroth dilution methods for testing antimicrobial compounds; J. Microbiol. Methods. 107 (2014), 98-105.
    (go to article)
  48. E. Słomińska, T. Borkowski, I. Rybakowska, M. Abramowicz-Glinka, Cz. Orlewska, R. Smolenski; In Vitro and Cellular Effects of 4-Pyridone-3-Carboxamide Riboside on Enzymes of Nucleotide Metabolism; Nucleos. Nucleot. Nucleic Acids. 33 (2014), 353-357.
    (go to article)
  49. J. Sławiński, Z. Brzozowski , B. Żołnowska, K. Szafrański, A. Pogorzelska, D. Vullo, C.T. Suipuran; Synthesis of a new series of N4-substituted 4-(2-aminoethyl)benzenesulfonamides and their inhibitory effect on human carbonic anhydrase cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII Eur. J. Med. Chem. 84 (2014), 59-67 (go to full text)
  50. J. Sławiński, A. Pogorzelska, B. Żołnowska, K. Brożewicz, D. Vullo, C.T. Suipuran Carbonic anhydrase inhibitors. Synthesis of a novel series of 5-substituted 2,4-dichlorobenzenesulfonamides and their inhibition of human cytosolic isozymes i and II and the transmembrane tumor-associated isozymes IX and XII Eur. J. Med. Chem. 82 (2014), 47-55 (full version)
  51. Z. Brzozowski, J. Sławiński, K. Szafrański On the reactioj products of 4-substituted 3-pyridinesulfonamides with some benzenesulfonyl chloride derivatives J. Heterocyclic Chem. 51 (2014), 11-17 (przejdź do artykułu)
  52. A. bogdanowicz, H. Foks, K. Gobis, A. Kędzia, E. Kwapisz, A. Olczak, M.L. Główka; The Synthesis and Antibacterial Activity of Novel 4-Pyrrolidin-3-cyanopyridine Derivatives; J. Het. Chem. 50 (2013), 544-550
    (go to article)
  53. J. Saczewski, M. Korcz, P. Karczewska, M. Gdaniec; Reactivity of cyclic alkoxyguanidines – experimental and theoretical studies; Arkivoc, part IV (2013), 346-362.
    (go to article)
  54. M. Belka, J. Slawinski, L. Konieczna, P. Kawczak, T. Ciesielski, T. Baczek; Antitumor Activity of Novel Benzensulfonamide Derivatives in View of their Physiochemical Properties Searched by Principal Component Analysis; Med. Chem. 9 (2013), 517-525 (go to article)
  55. J. Sławiński, K. Szafrański, D. Vullo, C.T. Supuran, Carbonic anhydrase inhibitors. Synthesis of heterocyclic 4-substituted pyridine-3-sulfonamide derivativesband their inhibition of the human cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII, Eur. J. Med. Chem. 69, (2013), 701-710 (go to article)
  56. Z. Brzozowski, J. Sławiński, Synthesis of Novel Series of 6-Chloro-1,1-dioxo-1,4,2-benzodithiazine derivatives with potential biological activity, J. Heterocyclic Chem., 50, 5, (2013) 1099–1107(go to article)
  57. J. Sławiński, A. Pogorzelska, B. Żołnowska, T. Laskowski, P. Sowiński, Synthesis and structure determination of 2,3-diaryl-9,9-dioxo-1H-9-thia-1,4,4a,7,10-pentaazaphenanthrene-2-ols, Tetrahedron 69 (2013) 8675-8679 (go to article)
  58. K. Gobis, H. Foks, J. Sławiński, E. Augustynowicz-Kopeć, A Napiórkowska, Synthesis and biological activity of novel 3-heteroaryl-2H-pyrido[4,3-e][1,2,4]thiadiazine and 3-heteroaryl-2H-benzo[e][1,2,4]thiadiazine 1,1-dioxides. Monatsh. Chem. 144, 8 (2013) 1197-1203 (go to article)
  59. Z. Brzozowski, B. Żołnowska, J. Sławiński, Synthesis of a new series of biologically interesting 6'-chloro-1',1'-dioxospiro[4H-benzo[d[1,3,7]oxadizocine-4,3'(2H)-[1,4,2]benzodithiazine-2,6(1H,5H)dione derivatives Monatsh. Chem. 144, 9 (2013) 1397-1405 (go to article)
  60. K. Gobis, H. Foks, J. Sławiński, A. Sikorski, D. Trzybiński, E. Augustynowicz-Kopeć, A Napiórkowska, K. Bojanowski, Synthesis, structure and biological activity of novel heterocyclic sulfonyl-carboximidamides. Monatsh. Chem. 144, 5 (2013) 647-658 (go to article)
  61. J. Sławiński, B. Żołnowska, D. Pirska, A. Kędzia, E. Kwapisz, Synthesis and antibacterial activity of novel 4-chloro-2-mercaptobenzenesulfonamide derivatives, J. Enzyme Inhib. Med. Chem. 28 (2013) 41-51 (go to article)
  62. J. Sławiński, B. Żołnowska, Cz. Orlewska, J. Chojnacki, Synthesis and molecular structure of novel 2-alkylthio-4-chloro-N -(5-oxo-4,5-dihydro-1H -1,2,4-triazolo-3-yl)-5-methylbenzenesulfonamides with potential anticancer activity Monatsh. Chem. 143, 12 (2012) 1705-1718 (go to article)
  63. Z. Brzozowski, J. Sławiński, D. Vullo, C.T. Supuran, Carbonic anhydrase inhibitors, regioselective synthesis of novel series 1-substituted 1,4-dihydro-4-oxo-3-pyridinesulfonamides and their inhibition of the human cytosolic isozymes I and II and transmembrane cancer associated isozymes IX and XII, Eur. J. Med. Chem. 56, (2012) 282-291
  64. K.Brożewicz, J. Sławiński, , 1-(2-Mercaptobenzenesulfonyl)-3-hydroxyguanidines – Novel potent antiproliferatives, synthesis and in vitro biological activity, Eur. J. Med. Chem . 55, (2012) 384-394
  65. K. Gobis, H. Foks, K. Wiśniewska, M. Dąbrowska-Szponar, E. Augustynowicz-Kopeć, A. Napiórkowska, Synthesis, and antimicrobal activity of novel heterocyclic sulfamoyl-phenyl-carboximidamides derived from clinically applied sulfonamides, Arch. Pharm. 345, 11 (2012) 911-917
  66. K. Gobis, H. Foks, K. Bojanowski E. Augustynowicz-Kopeć, A. Napiórkowska, Synthesis, of novel 3-cyclohexylpropanoic acid-derived nitrogen heterocyclic compounds and their evaluation for tuberculostatic activity. Bioorg. Med. Chem. 20, 1 (2012) 137-144
  67. K. Gobis, H. Foks, K. Wiśniewska, M. Dąbrowska-Szponar, E. Augustynowicz-Kopeć, A. Napiórkowska, A. Sikorski, Synthesis, structure, and antimicrobal activity of heterocyclic phenylsulfonyl- and 4-aminophenylsulfonyl-carboximidamides, Monatsh. Chem. 143, 8 (2012) 1161-1169
  68. K. Gobis, H. Foks, E. Augustynowicz-Kopeć, A. Napiórkowska, M. Szczesio, A. Olczak, M.L. Główka, Synthesis, characterization, and tuberculostatic activity of novel 2-(4-nitrobenzoyl)hydrazinecarbodithioic acid derivatives , Monatsh. Chem. 143, 4 (2012) 607-617
  69. K. Gobis, H. Foks, E. Augustynowicz-Kopeć, A. Napiórkowska; Synthesis and tuberculostatic activity of novel diverse heterocyclic compounds derived from heterocyclic carbohydrazides and methyl 2-heteroaroylhydrazinecarbodithioates, Heterocycles, 58, 4 (2012) 871–885
  70. K. Brożewicz, J. Sławiński, Synthesis and in vitro activity of novel 2-benzylthio-4-chloro-5-(1,3,4-oxadiazol-2-yl)benzenesulfonamide derivatives, Monatsh. Chem., 143, 6 (2012) 975-984
  71. Z. Brzozowski, J. Sławiński, M. Gdaniec, A. Innocenti, C.T. Supuran, Carbonic anhydrase inhibitors. Synthesis, molecular structures, and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with novel 3-pyridinesulfonamide derivatives, Eur. J. Med. Chem., 46, 9 (2011) 4403–4410
  72. J. Sławiński, K. Brożewicz, A. Fruziński, M.L. Główka, Synthesis and antitumor activity of novel N'-(2-benzylthiobenzenesulfonyl)-1H-pyrazole-1-amidine derivatives, Heterocycles, 83, 5 (2011) 1093–1109
  73. Z. Brzozowski, J. Sławiński, A. Innocenti, C.T. Supuran, Carbonic anhydrase inhibitors, regioselective synthesis of novel 1-substituted 1,4-dihydro-4-oxo-3-pyridinesulfonamides and their inhibition of the human cytosolic isozymes I and II and transmembrane cancer associated isozymes IX and XII, Eur. J. Med. Chem., 45, 9 (2010) 3656–3661
  74. Z. Brzozowski, J. Sławiński, F. Sączewski, A. Innocenti, C.T. Supuran, Carbonic anhydrase inhibitors: Synthesis and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with 4-substituted 3-pyridinesulfonamides, Eur. J. Med. Chem., 45, 6 (2010) 2396–2404
  75. Z. Brzozowski, J. Sławiński, Reaction products of activated aromatic and heteroaromatic chlorides with N,_N_-disubstituted formamides, Synth. Commun., 40 (2010) 1639–1645
  76. K. Gobis, H. Foks, Microwave-assisted synthesis of novel 4-N,N-dimethylamino- and 4-cycloamino- substituted 1,2,4-triazole-3-thiones, Heteroatom, 21, 3 (2010) 188–195
  77. B. Pilarski, A. Dobkowska, H. Foks, T. Michałowski, Modelling of acid-base equilibria in binary-solvent systems: a comparative study, Talanta, 80 (2010) 1073–1080
  78. Z. Brzozowski, J. Sławiński, A. Kędzia, E. Kwapisz, M. Gdaniec, Application of 3-methylthiopyrido[4,3-e]-1,4,2-dithiazine 1,1-dioxide to the synthesis of novel series of 4H-pyrido[4,3-e]-1,2,4-thiadiazine derivatives with potential biological activity, J. Heterocyclic Chem., 46, 6 (2009) 1396–1403
  79. Z. Brzozowski, F. Sączewski, J. Sławiński, T. Sanchez, N. Neamati, Synthesis and anti-HIV-1 integrase activities of 3-aroyl-2,3-dihydro-1,1-dioxo-1,4,2-benzodithiazines, Eur. J. Med. Chem., 44, 1 (2009) 190–196
  80. K. Gobis, H. Foks, A. Kędzia, M. Wierzbowska, Z. Zwolska, Synthesis and antibacterial activity of novel pyridine and pyrazine derivatives obtained from amidoximes, J. Heterocyclic Chem. , 46, 6 (2009) 1271–1279
  81. A. Bogdanowicz, H. Foks, A. Kędzia, E. Kwapisz, Z. Zwolska, E. Augustynowicz-Kopeć, The synthesis and microbiological activity of new 4-chloropyridin-2-yl derivatives, Heterocycles, 78, 9 (2009) 2217–2231
  82. H. Foks, K. Wisterowicz, A. Miszke, K. Brożewicz, K. Wiśniewska, M. Dąbrowska-Szponar, Synthesis, fungicidal and antibacterial activity of new pyridazine derivatives, Heterocycles, 78, 4 (2009) 961–975
  83. W. Konieczny, M. T. Konieczny, Synthesis of thioflavanone and flavanone derivatives by cyclization of chalcones, Synthesis, 11 (2009) 1811–1814
  84. M. T. Konieczny, Paweł Sowiński, Mechanism of isomerization and acid-induced transformations of 3'-hydroxy-4,4'-dimethoxy-3'-methyl-3-oxo-7,7'-bis(piperidinocarbonyloxy)-2,2-spirobi[2H,2'H,3H,3'H-benzo[b]thiophene]. Unusual equilibrium between the spiro and 3-hydroxybenzothiophene systems, Bull. Chem. Soc. Jpn., 82, 5 (2009) 600–602
  85. F. Sączewski, A. Innocenti, J. Sławiński, A. Kornicka, Z. Brzozowski, E. Pomarnacka, A. Scozzafava, C. Temperini, C. T. Supuran, Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with _S_-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides, Bioorg. Med. Chem., 16, 7 (2008) 3933–3940
  86. Z. Brzozowski, J. Sławiński, F. Sączewski, T. Sanchez, N. Neamati, Synthesis, anti-HIV-1 integrase, and cytotoxic activities of 4-chloro-N-(4-oxopyrimidin-2-yl)-2-mercaptobenzenesulfonamide derivatives, Eur. J. Med. Chem., 43 (2008) 1188–1198
  87. A. Miszke, H. Foks, K. Brożewicz, A. Kędzia, E. Kwapisz, Z. Zwolska, The synthesis and microbiological activity of 2-mercapto-4-methoxypyridine-3-carbonitrile derivatives, Heterocycles, 75, 11 (2008) 2723–2734
  88. Z. Brzozowski, F. Sączewski, J. Sławiński, Syntheses of potassium 1,1-dioxopyrido[4,3-e]-1,4,2-dithiazine-3-thiolate and its application to the synthesis of novel sulfonamides with potential biological activity, J. Heterocyclic Chem., 45, 5 (2008) 1407–1413
  89. B. Saraswathyamma, I. Grzybowska, C. Orlewska, J. Radecki, W. Dehaen, K. G. Kumar, H. Radecka, Electroactive dipyrromethene-Cu(II) monolayers deposited onto gold electrodes for voltammetric determination of paracetamol, Electroanalysis, 20, 21 (2008) 2317–2323
  90. I. Szymańska, M. Stobiecka, C. Orlewska, T. Rohand, D. Janssen, W. Dehaen, H. Radecka, Electroactive dipyrromethene – Cu(II) self-assembled monolayers: complexation reaction on the surface of gold electrodes, Langmuir, 24, 19 (2008) 11239–11245
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Krzysztof Szafrański